SYNTHESIS OF 3-CYANOBENZEN-1-SULFONYL CHLORIDES
Abstract and keywords
Abstract (English):
The paper presents a preparation method for 3-cyanobenzene-1-sulfonyl chlorides, valuable reagents for the fine organic synthesis used in the preparation of antiplatelet agents and agricultural germicides, pharmaceutical compositions, and biologically active compounds.

Keywords:
preparation method, 3-cyanobenzene-1-sulfonyl chlorides, antiplatelet agents, agricultural germicides
Text
Publication text (PDF): Read Download
References

1. Perzborn E., Seuter F., Fruchtmann R., Kohlsdorfer C. Substituted phenyl-sulphon amides: pat. DE3632329(A1) Germaniya. N 19863632329. opubl. 31.03.1988.

2. Igarashi K., Enomoto Y., Yanagida H., Gohara M., Iida N., Ozawa S., Kuwazuka T. Sulfonamide based compound and agricultural germicide: pat. JPH0655708 (B2) Yaponiya. N 19850099595. opubl. 27.07.1994.

3. Witte E.-C., Stegmeier K., Doerge L. Sulfonamidoalkyl cycloalkane compounds, processes for their production and pharmaceutical preparations: pat. DE3829455(A1) Germaniya. N 19883829455. opubl. 15.03.1990.

4. Witte E.-C., Stegmeier K., Dorge L., Doerge, L. Sulfonamidoalkyl cycloalkane compounds, processes for their production and pharmaceutical preparations: pat. EP0361113 (B1) Evropa. N 19890115912. opubl. 07.07.1993.

5. Owa T., Yoshino H., Okauchi T., et al. J. Med. Chem. 1999. V. 42. N. 19. P. 3789-3799.

6. Wakabayashi T., Ono N., Semba T., Haneda T. Antitumor agent comprising combination of sulfonamide-containing heterocyclic compound with an angiogenesis inhibitor: pat. US2005119303 (A1) SShA. N 20040504676. opubl. 02.06.2005.

7. Mrozik H. Anthelmintic substituted sulfonamide derivatives: zayavka US3953492 (A) SShA. N 19750562712. opubl. 27.04.1976.

8. Hagmann W., Lin L., Liu P., Mumford R., Reger T., Smith N., Stock N., Zunic J. Vla-4 antagonists: pat. US2007179190 (A1) SShA. N 20050591820. opubl. 02.08.2007.

9. Reger T.S., Zunic J., Stock N., et al. Bioorg. Med. Chem. Lett. 2010. V. 20. N. 3. P. 1173–1176.

10. Aldrich Chemistry 2012-2014: Handbook of Fine Chemicals. Sigma-Aldrich, 2011. R. 3216.

11. Dzhil'bert E.E. Sul'firovanie organicheskih soedineniy. Per. s angl. pod red. A.I. Gershenovicha. M.: Himiya, 1969. 416 s. Gilbert E.E. Sulfonation and related reactions. New York: Interscience Publishers, 1965. 529 p.

12. Cremlyn R.J. Chlorosulfonic acid: A versatile reagent. RSC Publishing, 2002. 322 p.

13. Malet-Sanz L., Ley S.V., Baxendale I.R., Madrzak J. Preparation of arylsulfonyl chlorides by chlorosulfonylation of in situ generated diazonium salts using a continuous flow reactor. Org. Biomol. Chem. 2010. N. 8. P. 5324-5332.

14. Tarasov A.V., Moskvichev Yu.A., Pisarev P.K., Nikiforova A.A. Sposob polucheniya arilhlorsul'fonilbenzamidov iz benzoynyh kislot: pat. RF № 2298548 C1. 10.05.2007.

15. Obschaya organicheskaya himiya. V 12 kn. Pod red. D. Barotna, U.D. Ollisa. Kn. 3. Azotsoderzhaschie soedineniya. M.: Himiya. 1982. 736 s. Comprehensive organic chemistry: The synthesis and reactions of organic compounds. A series of 6 volumes. Edited by D.Barton and W.D.Ollis. Volume 2. Nitrogen Compounds. Pergamon Press. 1979.

16. Harrison I.T., Harrison S. Compendium of Organic Synthetic Methods. John Wiley & Sons, Inc. 1971. 529 p.

Login or Create
* Forgot password?